# | Title | Journal | Year | Citations |
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1 | TMPRSS2 and furin are both essential for proteolytic activation of SARS-CoV-2 in human airway cells | Life Science Alliance | 2020 | 643 |
2 | Lipoxin and resolvin biosynthesis is dependent on 5‐lipoxygenase activating protein | FASEB Journal | 2015 | 73 |
3 | Structural Insights into Plasticity and Discovery of Remdesivir Metabolite GS-441524 Binding in SARS-CoV-2 Macrodomain | ACS Medicinal Chemistry Letters | 2021 | 35 |
4 | l-Thyroxin and the Nonclassical Thyroid Hormone TETRAC Are Potent Activators of PPARγ | Journal of Medicinal Chemistry | 2020 | 31 |
5 | Demonstrating Ligandability of the LC3A and LC3B Adapter Interface | Journal of Medicinal Chemistry | 2021 | 25 |
6 | Discovery of the First in Vivo Active Inhibitors of the Soluble Epoxide Hydrolase Phosphatase Domain | Journal of Medicinal Chemistry | 2019 | 21 |
7 | Michael acceptor containing drugs are a novel class of 5-lipoxygenase inhibitor targeting the surface cysteines C416 and C418 | Biochemical Pharmacology | 2017 | 19 |
8 | Heterodimer formation with retinoic acid receptor RXRα modulates coactivator recruitment by peroxisome proliferator-activated receptor PPARγ | Journal of Biological Chemistry | 2021 | 17 |
9 | Chiral chromatography–tandem mass spectrometry applied to the determination of pro-resolving lipid mediators | Journal of Chromatography A | 2014 | 16 |
10 | Exploring CYP2J2: lipid mediators, inhibitors and therapeutic implications | Drug Discovery Today | 2020 | 14 |
11 | Design, Synthesis, and Structure–Activity Relationship Studies of Dual Inhibitors of Soluble Epoxide Hydrolase and 5-Lipoxygenase | Journal of Medicinal Chemistry | 2020 | 13 |
12 | First Structure–Activity Relationship Study of Potent BLT2 Agonists as Potential Wound-Healing Promoters | Journal of Medicinal Chemistry | 2020 | 12 |
13 | Structure-Based Design of Dual Partial Peroxisome Proliferator-Activated Receptor γ Agonists/Soluble Epoxide Hydrolase Inhibitors | Journal of Medicinal Chemistry | 2021 | 10 |
14 | Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPARγ Modulation | Journal of the American Chemical Society | 2023 | 10 |
15 | Computer-Aided Selective Optimization of Side Activities of Talinolol | ACS Medicinal Chemistry Letters | 2019 | 9 |
16 | Systematic Assessment of Fragment Identification for Multitarget Drug Design | ChemMedChem | 2021 | 9 |
17 | Combined Cardioprotective and Adipocyte Browning Effects Promoted by the Eutomer of Dual sEH/PPARγ Modulator | Journal of Medicinal Chemistry | 2021 | 8 |
18 | Photosensitization enables Pauson-Khand–type reactions with nitrenes | Science | 2024 | 8 |
19 | AGMO Inhibitor Reduces 3T3-L1 Adipogenesis | Cells | 2021 | 6 |
20 | Structure optimization of a new class of PPARγ antagonists | Bioorganic and Medicinal Chemistry | 2019 | 5 |
21 | Discovery of Irbesartan Derivatives as BLT2 Agonists by Virtual Screening | ACS Medicinal Chemistry Letters | 2021 | 5 |
22 | Phenolate‐Induced N−O Bond Formation versus Tiemann‐Type Rearrangement for the Synthesis of 3‐Aminobenzisoxazoles and 2‐Aminobenzoxazoles | ChemistryOpen | 2022 | 4 |
23 | Development and Characterization of a Fluorescent Ligand for Leukotriene B4 Receptor 2 in Cells and Tissues | Journal of Medicinal Chemistry | 2022 | 3 |
24 | Photochemistry in Medicinal Chemistry and Chemical Biology | Journal of Medicinal Chemistry | 2024 | 2 |
25 | Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine‐Independent and Chronic Itch | Advanced Science | 2024 | 0 |
26 | Development of a Potent and Selective G2A (GPR132) Agonist | Journal of Medicinal Chemistry | 0 | 0 |
27 | A C-Degron Structure-Based Approach for the Development of Ligands Targeting the E3 Ligase TRIM7 | ACS Chemical Biology | 2024 | 0 |
28 | Structural Optimization of Oxaprozin for Selective Inverse Nurr1 Agonism | Journal of Medicinal Chemistry | 0 | 0 |
29 | SPMs exert anti-inflammatory and pro-resolving effects through positive allosteric modulation of the prostaglandin EP4 receptor | Proceedings of the National Academy of Sciences of the United States of America | 2024 | 0 |