| 1 | Protein and ligand preparation: parameters, protocols, and influence on virtual screening enrichments | Journal of Computer-Aided Molecular Design | 2013 | 5,333 |
| 2 | MOPAC: A semiempirical molecular orbital program | Journal of Computer-Aided Molecular Design | 1990 | 2,683 |
| 3 | Ligand docking and binding site analysis with PyMOL and Autodock/Vina | Journal of Computer-Aided Molecular Design | 2010 | 2,116 |
| 4 | Epik: a software program for pK a prediction and protonation state generation for drug-like molecules | Journal of Computer-Aided Molecular Design | 2007 | 1,877 |
| 5 | (null) | Journal of Computer-Aided Molecular Design | 1997 | 1,573 |
| 6 | Virtual Computational Chemistry Laboratory – Design and Description | Journal of Computer-Aided Molecular Design | 2005 | 1,355 |
| 7 | Molecular graph convolutions: moving beyond fingerprints | Journal of Computer-Aided Molecular Design | 2016 | 1,294 |
| 8 | (null) | Journal of Computer-Aided Molecular Design | 2002 | 1,123 |
| 9 | (null) | Journal of Computer-Aided Molecular Design | 2001 | 1,091 |
| 10 | PHASE: a new engine for pharmacophore perception, 3D QSAR model development, and 3D database screening: 1. Methodology and preliminary results | Journal of Computer-Aided Molecular Design | 2006 | 1,085 |
| 11 | Distributed automated docking of flexible ligands to proteins: Parallel applications of AutoDock 2.4 | Journal of Computer-Aided Molecular Design | 1996 | 954 |
| 12 | Towards the comprehensive, rapid, and accurate prediction of the favorable tautomeric states of drug-like molecules in aqueous solution | Journal of Computer-Aided Molecular Design | 2010 | 894 |
| 13 | The development of a simple empirical scoring function to estimate the binding constant for a protein-ligand complex of known three-dimensional structure | Journal of Computer-Aided Molecular Design | 1994 | 893 |
| 14 | The computer program LUDI: A new method for the de novo design of enzyme inhibitors | Journal of Computer-Aided Molecular Design | 1992 | 779 |
| 15 | VEGA – An open platform to develop chemo-bio-informatics applications, using plug-in architecture and script programming | Journal of Computer-Aided Molecular Design | 2004 | 671 |
| 16 | PRODRG, a program for generating molecular topologies and unique molecular descriptors from coordinates of small molecules | Journal of Computer-Aided Molecular Design | 1996 | 663 |
| 17 | (null) | Journal of Computer-Aided Molecular Design | 2003 | 645 |
| 18 | Online chemical modeling environment (OCHEM): web platform for data storage, model development and publishing of chemical information | Journal of Computer-Aided Molecular Design | 2011 | 603 |
| 19 | (null) | Journal of Computer-Aided Molecular Design | 2002 | 584 |
| 20 | Interpretation of machine learning models using shapley values: application to compound potency and multi-target activity predictions | Journal of Computer-Aided Molecular Design | 2020 | 578 |
| 21 | MAB, a generally applicable molecular force field for structure modelling in medicinal chemistry | Journal of Computer-Aided Molecular Design | 1995 | 569 |
| 22 | Computer-aided drug design platform using PyMOL | Journal of Computer-Aided Molecular Design | 2010 | 557 |
| 23 | Scoring noncovalent protein-ligand interactions: A continuous differentiable function tuned to compute binding affinities | Journal of Computer-Aided Molecular Design | 1996 | 556 |
| 24 | Local elevation: A method for improving the searching properties of molecular dynamics simulation | Journal of Computer-Aided Molecular Design | 1994 | 551 |
| 25 | Surflex-Dock 2.1: Robust performance from ligand energetic modeling, ring flexibility, and knowledge-based search | Journal of Computer-Aided Molecular Design | 2007 | 540 |
| 26 | Testing and validation of the Automated Topology Builder (ATB) version 2.0: prediction of hydration free enthalpies | Journal of Computer-Aided Molecular Design | 2014 | 479 |
| 27 | Estimation of the size of drug-like chemical space based on GDB-17 data | Journal of Computer-Aided Molecular Design | 2013 | 471 |
| 28 | FRED and HYBRID docking performance on standardized datasets | Journal of Computer-Aided Molecular Design | 2012 | 466 |
| 29 | Guidelines for the analysis of free energy calculations | Journal of Computer-Aided Molecular Design | 2015 | 461 |
| 30 | (null) | Journal of Computer-Aided Molecular Design | 1998 | 427 |
| 31 | LUDI: rule-based automatic design of new substituents for enzyme inhibitor leads | Journal of Computer-Aided Molecular Design | 1992 | 419 |
| 32 | FreeSolv: a database of experimental and calculated hydration free energies, with input files | Journal of Computer-Aided Molecular Design | 2014 | 412 |
| 33 | (null) | Journal of Computer-Aided Molecular Design | 2002 | 410 |
| 34 | Variability in docking success rates due to dataset preparation | Journal of Computer-Aided Molecular Design | 2012 | 403 |
| 35 | Development and validation of a modular, extensible docking program: DOCK 5 | Journal of Computer-Aided Molecular Design | 2006 | 398 |
| 36 | TargetNet: a web service for predicting potential drug–target interaction profiling via multi-target SAR models | Journal of Computer-Aided Molecular Design | 2016 | 374 |
| 37 | Evaluation of the performance of 3D virtual screening protocols: RMSD comparisons, enrichment assessments, and decoy selection—What can we learn from earlier mistakes? | Journal of Computer-Aided Molecular Design | 2008 | 373 |
| 38 | A fast new approach to pharmacophore mapping and its application to dopaminergic and benzodiazepine agonists | Journal of Computer-Aided Molecular Design | 1993 | 368 |
| 39 | A genetic algorithm for flexible molecular overlay and pharmacophore elucidation | Journal of Computer-Aided Molecular Design | 1995 | 356 |
| 40 | Boltzmann's principle, knowledge-based mean fields and protein folding. An approach to the computational determination of protein structures | Journal of Computer-Aided Molecular Design | 1993 | 355 |
| 41 | Docking and scoring with ICM: the benchmarking results and strategies for improvement | Journal of Computer-Aided Molecular Design | 2012 | 349 |
| 42 | Sample-distance partial least squares: PLS optimized for many variables, with application to CoMFA | Journal of Computer-Aided Molecular Design | 1993 | 347 |
| 43 | (null) | Journal of Computer-Aided Molecular Design | 2002 | 334 |
| 44 | Class IV charge models: A new semiempirical approach in quantum chemistry | Journal of Computer-Aided Molecular Design | 1995 | 320 |
| 45 | AM1-SM2 and PM3-SM3 parameterized SCF solvation models for free energies in aqueous solution | Journal of Computer-Aided Molecular Design | 1992 | 319 |
| 46 | Comparative study of several algorithms for flexible ligand docking | Journal of Computer-Aided Molecular Design | 2003 | 319 |
| 47 | Lessons learned from comparing molecular dynamics engines on the SAMPL5 dataset | Journal of Computer-Aided Molecular Design | 2016 | 318 |
| 48 | Strategic approaches to drug design. I. An integrated software framework for molecular modelling | Journal of Computer-Aided Molecular Design | 1987 | 314 |
| 49 | HINT: A new method of empirical hydrophobic field calculation for CoMFA | Journal of Computer-Aided Molecular Design | 1991 | 313 |
| 50 | Recommendations for evaluation of computational methods | Journal of Computer-Aided Molecular Design | 2008 | 308 |