# | Title | Journal | Year | Citations |
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1 | Protein and ligand preparation: parameters, protocols, and influence on virtual screening enrichments | Journal of Computer-Aided Molecular Design | 2013 | 4,278 |
2 | Molden: a pre- and post-processing program for molecular and electronic structures | Journal of Computer-Aided Molecular Design | 2000 | 2,851 |
3 | MOPAC: A semiempirical molecular orbital program | Journal of Computer-Aided Molecular Design | 1990 | 2,572 |
4 | Ligand docking and binding site analysis with PyMOL and Autodock/Vina | Journal of Computer-Aided Molecular Design | 2010 | 1,566 |
5 | Epik: a software program for pK a prediction and protonation state generation for drug-like molecules | Journal of Computer-Aided Molecular Design | 2007 | 1,564 |
6 | Empirical scoring functions: I. The development of a fast empirical scoring function to estimate the binding affinity of ligands in receptor complexes | Journal of Computer-Aided Molecular Design | 1997 | 1,517 |
7 | Virtual Computational Chemistry Laboratory – Design and Description | Journal of Computer-Aided Molecular Design | 2005 | 1,270 |
8 | Molecular graph convolutions: moving beyond fingerprints | Journal of Computer-Aided Molecular Design | 2016 | 1,056 |
9 | DOCK 4.0: search strategies for automated molecular docking of flexible molecule databases | Journal of Computer-Aided Molecular Design | 2001 | 1,040 |
10 | Further development and validation of empirical scoring functions for structure-based binding affinity prediction | Journal of Computer-Aided Molecular Design | 2002 | 1,036 |
11 | PHASE: a new engine for pharmacophore perception, 3D QSAR model development, and 3D database screening: 1. Methodology and preliminary results | Journal of Computer-Aided Molecular Design | 2006 | 983 |
12 | Distributed automated docking of flexible ligands to proteins: Parallel applications of AutoDock 2.4 | Journal of Computer-Aided Molecular Design | 1996 | 916 |
13 | The development of a simple empirical scoring function to estimate the binding constant for a protein-ligand complex of known three-dimensional structure | Journal of Computer-Aided Molecular Design | 1994 | 874 |
14 | Towards the comprehensive, rapid, and accurate prediction of the favorable tautomeric states of drug-like molecules in aqueous solution | Journal of Computer-Aided Molecular Design | 2010 | 796 |
15 | The computer program LUDI: A new method for the de novo design of enzyme inhibitors | Journal of Computer-Aided Molecular Design | 1992 | 752 |
16 | VEGA – An open platform to develop chemo-bio-informatics applications, using plug-in architecture and script programming | Journal of Computer-Aided Molecular Design | 2004 | 646 |
17 | PRODRG, a program for generating molecular topologies and unique molecular descriptors from coordinates of small molecules | Journal of Computer-Aided Molecular Design | 1996 | 613 |
18 | Rational selection of training and test sets for the development of validated QSAR models | Journal of Computer-Aided Molecular Design | 2003 | 600 |
19 | A review of protein-small molecule docking methods | Journal of Computer-Aided Molecular Design | 2002 | 565 |
20 | Property distribution of drug-related chemical databases | Journal of Computer-Aided Molecular Design | 2000 | 552 |
21 | MAB, a generally applicable molecular force field for structure modelling in medicinal chemistry | Journal of Computer-Aided Molecular Design | 1995 | 548 |
22 | Scoring noncovalent protein-ligand interactions: A continuous differentiable function tuned to compute binding affinities | Journal of Computer-Aided Molecular Design | 1996 | 545 |
23 | Surflex-Dock 2.1: Robust performance from ligand energetic modeling, ring flexibility, and knowledge-based search | Journal of Computer-Aided Molecular Design | 2007 | 525 |
24 | Local elevation: A method for improving the searching properties of molecular dynamics simulation | Journal of Computer-Aided Molecular Design | 1994 | 521 |
25 | Online chemical modeling environment (OCHEM): web platform for data storage, model development and publishing of chemical information | Journal of Computer-Aided Molecular Design | 2011 | 479 |
26 | QXP: powerful, rapid computer algorithms for structure-based drug design | Journal of Computer-Aided Molecular Design | 1997 | 469 |
27 | Fast prediction and visualization of protein binding pockets with PASS | Journal of Computer-Aided Molecular Design | 2000 | 466 |
28 | Computer-aided drug design platform using PyMOL | Journal of Computer-Aided Molecular Design | 2011 | 445 |
29 | Testing and validation of the Automated Topology Builder (ATB) version 2.0: prediction of hydration free enthalpies | Journal of Computer-Aided Molecular Design | 2014 | 436 |
30 | FRED and HYBRID docking performance on standardized datasets | Journal of Computer-Aided Molecular Design | 2012 | 413 |
31 | LUDI: rule-based automatic design of new substituents for enzyme inhibitor leads | Journal of Computer-Aided Molecular Design | 1992 | 412 |
32 | Ligand binding affinity prediction by linear interaction energy methods | Journal of Computer-Aided Molecular Design | 1998 | 408 |
33 | Predictive QSAR modeling based on diversity sampling of experimental datasets for the training and test set selection | Journal of Computer-Aided Molecular Design | 2002 | 400 |
34 | Guidelines for the analysis of free energy calculations | Journal of Computer-Aided Molecular Design | 2015 | 398 |
35 | Prediction of binding constants of protein ligands: a fast method for the prioritization of hits obtained from de novo design or 3D database search programs | Journal of Computer-Aided Molecular Design | 1998 | 397 |
36 | Development and validation of a modular, extensible docking program: DOCK 5 | Journal of Computer-Aided Molecular Design | 2006 | 375 |
37 | A fast new approach to pharmacophore mapping and its application to dopaminergic and benzodiazepine agonists | Journal of Computer-Aided Molecular Design | 1993 | 364 |
38 | Estimation of the size of drug-like chemical space based on GDB-17 data | Journal of Computer-Aided Molecular Design | 2013 | 363 |
39 | Variability in docking success rates due to dataset preparation | Journal of Computer-Aided Molecular Design | 2012 | 358 |
40 | A genetic algorithm for flexible molecular overlay and pharmacophore elucidation | Journal of Computer-Aided Molecular Design | 1995 | 350 |
41 | Boltzmann's principle, knowledge-based mean fields and protein folding. An approach to the computational determination of protein structures | Journal of Computer-Aided Molecular Design | 1993 | 349 |
42 | Evaluation of the performance of 3D virtual screening protocols: RMSD comparisons, enrichment assessments, and decoy selection—What can we learn from earlier mistakes? | Journal of Computer-Aided Molecular Design | 2008 | 344 |
43 | Sample-distance partial least squares: PLS optimized for many variables, with application to CoMFA | Journal of Computer-Aided Molecular Design | 1993 | 341 |
44 | AM1-SM2 and PM3-SM3 parameterized SCF solvation models for free energies in aqueous solution | Journal of Computer-Aided Molecular Design | 1992 | 317 |
45 | Maximum common subgraph isomorphism algorithms for the matching of chemical structures | Journal of Computer-Aided Molecular Design | 2002 | 315 |
46 | FreeSolv: a database of experimental and calculated hydration free energies, with input files | Journal of Computer-Aided Molecular Design | 2014 | 313 |
47 | Strategic approaches to drug design. I. An integrated software framework for molecular modelling | Journal of Computer-Aided Molecular Design | 1987 | 311 |
48 | Class IV charge models: A new semiempirical approach in quantum chemistry | Journal of Computer-Aided Molecular Design | 1995 | 311 |
49 | HINT: A new method of empirical hydrophobic field calculation for CoMFA | Journal of Computer-Aided Molecular Design | 1991 | 306 |
50 | Comparative study of several algorithms for flexible ligand docking | Journal of Computer-Aided Molecular Design | 2003 | 304 |