| # | Title | Journal | Year | Citations |
|---|
| 1 | Synthesis, structure and anticancer activity of novel 2,4-diamino-1,3,5-triazine derivatives | European Journal of Medicinal Chemistry | 2006 | 80 |
| 2 | Synthesis and antibacterial activity of 1H-pyrazolo[3,4-b]pyrazine and -pyridine derivatives | Il Farmaco | 2005 | 75 |
| 3 | Modifications of quinolones and fluoroquinolones: hybrid compounds and dual-action molecules | Monatshefte Für Chemie | 2018 | 74 |
| 4 | Carbonic anhydrase inhibitors. Synthesis, and molecular structure of novel series N-substituted N′-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)guanidines and their inhibition of human cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII | European Journal of Medicinal Chemistry | 2014 | 61 |
| 5 | Synthesis and biological evaluation of hybrid quinolone-based quaternary ammonium antibacterial agents | European Journal of Medicinal Chemistry | 2019 | 53 |
| 6 | Acid-catalyzed synthesis of oxathiolone fused chalcones. Comparison of their activity toward various microorganisms and human cancer cells line | European Journal of Medicinal Chemistry | 2007 | 51 |
| 7 | Novel 2-benzylthio-5-(1,3,4-oxadiazol-2-yl)benzenesulfonamides with anticancer activity: Synthesis, QSAR study, and metabolic stability | European Journal of Medicinal Chemistry | 2017 | 50 |
| 8 | Electroactive Dipyrromethene‐Cu(II) Monolayers Deposited onto Gold Electrodes for Voltammetric Determination of Paracetamol | Electroanalysis | 2008 | 47 |
| 9 | Synthesis of Isomeric, Oxathiolone Fused Chalcones, and Comparison of Their Activity toward Various Microorganisms and Human Cancer Cells Line | Chemical and Pharmaceutical Bulletin | 2007 | 46 |
| 10 | Synthesis and evaluation of in vitro antimycobacterial activity of novel 1H-benzo[d]imidazole derivatives and analogues | European Journal of Medicinal Chemistry | 2015 | 44 |
| 11 | Active Benzimidazole Derivatives Targeting the MmpL3 Transporter in Mycobacterium abscessus | ACS Infectious Diseases | 2020 | 44 |
| 12 | Pharmacological Potential and Synthetic Approaches of Imidazo[4,5-b]pyridine and Imidazo[4,5-c]pyridine Derivatives | Molecules | 2017 | 41 |
| 13 | Carbonic anhydrase inhibitors. Synthesis of heterocyclic 4-substituted pyridine-3-sulfonamide derivatives and their inhibition of the human cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII | European Journal of Medicinal Chemistry | 2013 | 37 |
| 14 | Cysteine cathepsins as a prospective target for anticancer therapies—current progress and prospects | Biochimie | 2018 | 35 |
| 15 | Some reactions of 2-cyanomethylimidazo[4,5-b]pyridine with isothiocyanates. Antituberculotic activity of the obtained compounds | Die Pharmazie | 1998 | 35 |
| 16 | A Novel Nucleotide Found in Human Erythrocytes, 4-Pyridone-3-carboxamide-1-β-d-ribonucleoside Triphosphate* | Journal of Biological Chemistry | 2006 | 33 |
| 17 | Modelling of acid–base equilibria in binary-solvent systems: A comparative study | Talanta | 2010 | 28 |
| 18 | Rational design, synthesis and biological evaluation of thiadiazinoacridines: A new class of antitumor agents | Bioorganic and Medicinal Chemistry | 2003 | 27 |
| 19 | Synthesis and Tuberculostatic Activity of Some 2-Piperazinmethylene Derivatives 1,2,4-Triazole-3-Thiones | Phosphorus, Sulfur and Silicon and the Related Elements | 2005 | 27 |
| 20 | Synthesis and tuberculostatic activity of new benzimidazole derivatives | Chemistry of Heterocyclic Compounds | 2006 | 27 |
| 21 | Synthesis of novel 3-cyclohexylpropanoic acid-derived nitrogen heterocyclic compounds and their evaluation for tuberculostatic activity | Bioorganic and Medicinal Chemistry | 2012 | 27 |
| 22 | Novel 2-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)-1-(1,3,5-triazin-2-ylamino)guanidine derivatives: Inhibition of human carbonic anhydrase cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII, anticancer activity, and molecular modeling studies | European Journal of Medicinal Chemistry | 2018 | 26 |
| 23 | Lipophilicity Determination of Quaternary (Fluoro)Quinolones by Chromatographic and Theoretical Approaches | International Journal of Molecular Sciences | 2019 | 26 |
| 24 | Carbonic anhydrase inhibitors. Regioselective synthesis of novel 1-substituted 1,4-dihydro-4-oxo-3-pyridinesulfonamides and their inhibition of the human cytosolic isozymes I and II and transmembrane cancer-associated isozymes IX and XII | European Journal of Medicinal Chemistry | 2010 | 25 |
| 25 | 1 H -Benzo[ d ]Imidazole Derivatives Affect MmpL3 in Mycobacterium tuberculosis | Antimicrobial Agents and Chemotherapy | 2019 | 25 |
| 26 | New domino reaction. One pot synthesis of 4,7-dihydroxythioaurone derivatives from benzaldehydes and 4-acetyl-2-oxo-benz[1,3]oxathiole | Tetrahedron | 2005 | 23 |
| 27 | Structural factors affecting affinity of cytotoxic oxathiole-fused chalcones toward tubulin | European Journal of Medicinal Chemistry | 2015 | 23 |
| 28 | Hybrid Molecules Composed of 2,4-Diamino-1,3,5-triazines and 2-Imino-Coumarins and Coumarins. Synthesis and Cytotoxic Properties | Molecules | 2018 | 23 |
| 29 | Novel 2-(2-phenalkyl)-1H-benzo[d]imidazoles as antitubercular agents. Synthesis, biological evaluation and structure–activity relationship | Bioorganic and Medicinal Chemistry | 2015 | 22 |
| 30 | Is planarity of pyridin-2-yl- and pyrazin-2-yl-formamide thiosemicarbazones related to their tuberculostatic activity? X-ray structures of two pyrazine-2-carboxamide-N′-carbonothioyl-hydrazones | Journal of Molecular Structure | 2007 | 21 |
| 31 | (null) | Chemistry of Heterocyclic Compounds | 2002 | 19 |
| 32 | Synthesis and molecular structure of novel 2-(alkylthio)-4-chloro-N-(4,5-dihydro-5-oxo-1H-1,2,4-triazol-3-yl)-5-methylbenzenesulfonamides with potential anticancer activity | Monatshefte Für Chemie | 2012 | 18 |
| 33 | Comparison of fluorescence optical respirometry and microbroth dilution methods for testing antimicrobial compounds | Journal of Microbiological Methods | 2014 | 18 |
| 34 | Carbonic anhydrase inhibitors. Synthesis of a novel series of 5-substituted 2,4-dichlorobenzenesulfonamides and their inhibition of human cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII | European Journal of Medicinal Chemistry | 2014 | 18 |
| 35 | Synthesis and some reactions of 2-acetylimidazo[4,5-b]pyridine. Antituberculotic activity of the obtained compounds | Die Pharmazie | 1999 | 18 |
| 36 | Metabolism of 4-Pyridone-3-Carboxamide-1-ß-D- Ribonucleoside Triphosphate and Its Nucleoside Precursor in the Erythrocytes | Nucleosides, Nucleotides and Nucleic Acids | 2008 | 17 |
| 37 | Synthesis of a new series of N4-substituted 4-(2-aminoethyl)benzenesulfonamides and their inhibitory effect on human carbonic anhydrase cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII | European Journal of Medicinal Chemistry | 2014 | 17 |
| 38 | Novel 2-(2-alkylthiobenzenesulfonyl)-3-(phenylprop-2-ynylideneamino)guanidine derivatives as potent anticancer agents – Synthesis, molecular structure, QSAR studies and metabolic stability | European Journal of Medicinal Chemistry | 2017 | 17 |
| 39 | Antifungal action of the oxathiolone‐fused chalcone derivative | Mycoses | 2011 | 16 |
| 40 | 1-(2-Mercaptobenzenesulfonyl)-3-hydroxyguanidines – Novel potent antiproliferatives, synthesis and in vitro biological activity | European Journal of Medicinal Chemistry | 2012 | 16 |
| 41 | Novel 5-Substituted 2-(Aylmethylthio)-4-chloro-N-(5-aryl-1,2,4-triazin-3-yl)benzenesulfonamides: Synthesis, Molecular Structure, Anticancer Activity, Apoptosis-Inducing Activity and Metabolic Stability | Molecules | 2016 | 16 |
| 42 | Anticancer and antimicrobial activity of new copper (II) complexes | Journal of Inorganic Biochemistry | 2023 | 16 |
| 43 | Chemosensitization of multidrug resistant Candida albicans by the oxathiolone fused chalcone derivatives | Frontiers in Microbiology | 2015 | 15 |
| 44 | Experimental and theoretical studies on the tautomerism and reactivity of isoxazolo[3,4-b]quinolin-3(1H)-ones | Tetrahedron | 2015 | 15 |
| 45 | Synthesis and Tuberculostatic Activity Evaluation of Novel Benzazoles with Alkyl, Cycloalkyl or Pyridine Moiety | Molecules | 2018 | 15 |
| 46 | Studies on pyrazine derivatives. XXXIII. Synthesis and tuberculostatic activity of 1-[1-(2-pyrazinyl)-ethyl]-4-N-substituted thiosemicarbazide derivatives | Acta Poloniae Pharmaceutica | 1999 | 15 |
| 47 | Synthesis and tuberculostatic activity of some (4-phenylpiperazin-1-ylmethyl)-1,3,4-oxadiazole and (4-phenylpiperazin-1-ylmethyl)-1,2,4-triazole derivatives | Acta Poloniae Pharmaceutica | 2004 | 15 |
| 48 | Synthesis and Antibacterial Activity of Substituted Thiosemicarbazides and of 1,3,4-Thiadiazole or 1,2,4-Triazole Derivatives | Phosphorus, Sulfur and Silicon and the Related Elements | 2006 | 14 |
| 49 | Structural Factors Affecting Cytotoxic Activity of (E)‐1‐(Benzo[d ][1,3]oxathiol‐6‐yl)‐3‐phenylprop‐2‐en‐1‐one Derivatives | Chemical Biology and Drug Design | 2014 | 14 |
| 50 | Transfer of SAR information from hypotensive indazole to indole derivatives acting at α-adrenergic receptors: In vitro and in vivo studies | European Journal of Medicinal Chemistry | 2016 | 14 |
