| # | Title | Journal | Year | Citations |
|---|
| 1 | Molecular hybrids: A five-year survey on structures of multiple targeted hybrids of protein kinase inhibitors for cancer therapy | European Journal of Medicinal Chemistry | 2021 | 52 |
| 2 | Asymmetric Synthesis of Tailor-Made Amino Acids Using Chiral Ni(II) Complexes of Schiff Bases. An Update of the Recent Literature | Molecules | 2020 | 40 |
| 3 | Tailor-made amino acids in the design of small-molecule blockbuster drugs | European Journal of Medicinal Chemistry | 2021 | 31 |
| 4 | Nitric oxide protects against ferroptosis by aborting the lipid peroxidation chain reaction | Nitric Oxide - Biology and Chemistry | 2021 | 28 |
| 5 | Synthesis and evaluation of phenylisoserine derivatives for the SARS-CoV 3CL protease inhibitor | Bioorganic and Medicinal Chemistry Letters | 2017 | 24 |
| 6 | Tailor-made amino acid-derived pharmaceuticals approved by the FDA in 2019 | Amino Acids | 2020 | 24 |
| 7 | Design, synthesis and evaluation of curcumin-based fluorescent probes to detect Aβ fibrils | Bioorganic and Medicinal Chemistry Letters | 2018 | 21 |
| 8 | New pharmaceuticals approved by FDA in 2020: Small‐molecule drugs derived from amino acids and related compounds | Chirality | 2022 | 20 |
| 9 | Design and synthesis of a series of serine derivatives as small molecule inhibitors of the SARS coronavirus 3CL protease | Bioorganic and Medicinal Chemistry | 2016 | 19 |
| 10 | γ-Glutamylcysteine synthetase and γ-glutamyl transferase as differential enzymatic sources of γ-glutamylpeptides in mice | Amino Acids | 2020 | 15 |
| 11 | Structure activity relationship study of burkholdine analogues toward simple antifungal agents | Bioorganic and Medicinal Chemistry Letters | 2015 | 12 |
| 12 | Kitamura Electrophilic Fluorination Using HF as a Source of Fluorine | Molecules | 2020 | 12 |
| 13 | Synthesis and antifungal activities of cyclic octa-lipopeptide burkholdine analogues | Bioorganic and Medicinal Chemistry Letters | 2013 | 11 |
| 14 | Carnosine dipeptidase II (CNDP2) protects cells under cysteine insufficiency by hydrolyzing glutathione-related peptides | Free Radical Biology and Medicine | 2021 | 11 |
| 15 | Quantitative analysis of γ-glutamylpeptides by liquid chromatography-mass spectrometry and application for γ-glutamyltransferase assays | Analytical Biochemistry | 2019 | 10 |
| 16 | Michael addition reactions of chiral glycine Schiff base Ni (II)‐complex with 1‐(1‐phenylsulfonyl)benzene | Chirality | 2020 | 7 |
| 17 | Peptidomimetics and Peptide-Based Blockbuster Drugs | Current Organic Chemistry | 2021 | 7 |
| 18 | Synthetic study of peptide aldehyde via acetal/thioacetal transformation: application for Lys/Ser-containing peptides | Tetrahedron | 2015 | 6 |
| 19 | Fmoc-OPhth, the reagent of Fmoc protection | Tetrahedron Letters | 2017 | 6 |
| 20 | Synthesis of a secretoglobin 3A2 type C (98–139) fragment by Dawson’s native chemical ligation | Tetrahedron Letters | 2017 | 6 |
| 21 | Synthesis of a burkholdine analogue containing β-hydroxytyrosine | Bioscience, Biotechnology and Biochemistry | 2019 | 6 |
| 22 | Asymmetric Synthesis of α‐Difluorinated β‐Amino Sulfones through Detrifluoroacetylative Mannich Reactions | European Journal of Organic Chemistry | 2021 | 6 |
| 23 | Synthetic studies on homophymine B: solid phase synthesis of a cyclic fragment | Tetrahedron Letters | 2015 | 5 |
| 24 | Asymmetric Mannich reactions of (S)-N-tert-butylsulfinyl-3,3,3-trifluoroacetaldimines with yne nucleophiles | Beilstein Journal of Organic Chemistry | 2020 | 5 |
| 25 | Asymmetric Synthesis of N ‐Fmoc‐( S )‐7‐aza‐tryptophan via Alkylation of Chiral Nucleophilic Glycine Equivalent | European Journal of Organic Chemistry | 2021 | 5 |
| 26 | Aerobic oxidation of aldehydes to acids with N-hydroxyphthalimide derivatives | Tetrahedron Letters | 2021 | 5 |
| 27 | Asymmetric synthesis of ( S )‐3‐methyleneglutamic acid and its N ‐Fmoc derivative via Michael addition–elimination reaction of chiral glycine Ni (II) complex with enol tosylates | Chirality | 2021 | 5 |
| 28 | Synthesis of Bioactive Natural Products as Protein Inhibitors | Bioscience, Biotechnology and Biochemistry | 2012 | 4 |
| 29 | Synthesis of fully protected (2 R ,3 R ,4 S )-4-amino-7-guanidino-2,3-dihydroxy heptanoic acid | Tetrahedron Letters | 2017 | 4 |
| 30 | Design, Synthesis, Molecular Modeling and Biological Evaluation of Novel 1,5-Diarylpyrazole Carboxamide Derivatives as Antiproliferative Agents | Journal of Advanced Biomedical and Pharmaceutical Sciences | 2021 | 2 |
| 31 | Comparative study of different chiral ligands for dynamic kinetic resolution of amino acids | Chirality | 2021 | 1 |
| 32 | Design, synthesis, molecular docking and biological evaluation of novel 1,5-diarylpyrazole-N,O-dimethyl hydroxamate derivatives as antiproliferative agents. | Journal of Advanced Biomedical and Pharmaceutical Sciences | 2021 | 1 |
| 33 | The Hydrophobicity and Antifungal Potentiation of Burkholdine Analogues | Molecules | 2022 | 1 |
| 34 | Synthesis and Configuration Confirmation of the ATHOD Fatty Amino Acid Residue in the Burkholdines | Journal of Natural Products | 2022 | 1 |
