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Topics in Medicinal Chemistry
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top-articles
Topics in Medicinal Chemistry
0.4
(top 50%)
impact factor
326
(top 50%)
papers
1.1K
(top 50%)
citations
12
(top 50%)
h
-index
0.4
(top 50%)
extended IF
370
all documents
1.2K
doc citations
19
(top 50%)
g
-index
Top Articles
#
Title
Journal
Year
Citations
1
Targeting the MDM2-p53 Protein-Protein Interaction for New Cancer Therapeutics
Topics in Medicinal Chemistry
2012
60
2
Sideromycins as Pathogen-Targeted Antibiotics
Topics in Medicinal Chemistry
2017
44
3
The Influence of Bioisosteres in Drug Design: Tactical Applications to Address Developability Problems
Topics in Medicinal Chemistry
2013
30
4
Drug Design Based on the Carbon/Silicon Switch Strategy
Topics in Medicinal Chemistry
2014
25
5
Nanoparticles as Blood–Brain Barrier Permeable CNS Targeted Drug Delivery Systems
Topics in Medicinal Chemistry
2013
22
6
Tactics in Contemporary Drug Design
Topics in Medicinal Chemistry
2015
18
7
The Medicinal Chemistry of Tuberculosis Chemotherapy
Topics in Medicinal Chemistry
2011
17
8
Iminosugars: Therapeutic Applications and Synthetic Considerations
Topics in Medicinal Chemistry
2014
15
9
The Design, Development, and Evaluation of BACE1 Inhibitors for the Treatment of Alzheimer’s Disease
Topics in Medicinal Chemistry
2016
14
10
Past, Present, and Future of Antifungal Drug Development
Topics in Medicinal Chemistry
2016
14
11
Physical Properties in Drug Design
Topics in Medicinal Chemistry
2014
13
12
Viral RNA Targets and Their Small Molecule Ligands
Topics in Medicinal Chemistry
2017
13
13
Discovery and Application of FimH Antagonists
Topics in Medicinal Chemistry
2014
12
14
Approaches for the Discovery of Small Molecule Ligands Targeting microRNAs
Topics in Medicinal Chemistry
2017
12
15
Atypical Dopamine Uptake Inhibitors that Provide Clues About Cocaine's Mechanism at the Dopamine Transporter
Topics in Medicinal Chemistry
2008
11
16
Phosphodiesterase Inhibition to Target the Synaptic Dysfunction in Alzheimer’s Disease
Topics in Medicinal Chemistry
2010
11
17
Silicon Mimics of Unstable Carbon
Topics in Medicinal Chemistry
2014
11
18
The Oxazolidinones
Topics in Medicinal Chemistry
2017
11
19
Synergistic Antibiotic Combinations
Topics in Medicinal Chemistry
2017
11
20
The Antibiotic Future
Topics in Medicinal Chemistry
2017
11
21
Discovering New Medicines to Control and Eradicate Malaria
Topics in Medicinal Chemistry
2011
10
22
Selective and Dual Targeting of CCR2 and CCR5 Receptors: A Current Overview
Topics in Medicinal Chemistry
2014
10
23
Quorum Sensing Inhibitors as Pathoblockers for Pseudomonas aeruginosa Infections: A New Concept in Anti-Infective Drug Discovery
Topics in Medicinal Chemistry
2017
10
24
Relativistic Quantum Chemical and Molecular Dynamics Techniques for Medicinal Chemistry of Bioinorganic Compounds
Topics in Medicinal Chemistry
2021
10
25
Novel Small-Molecule Inhibitors of Src Kinase for Cancer Therapy
Topics in Medicinal Chemistry
2007
9
26
HDAC Inhibition in Cancer Therapy: An Increasingly Intriguing Tale of Chemistry, Biology and Clinical Benefit
Topics in Medicinal Chemistry
2007
9
27
The Discovery of Navitoclax, a Bcl-2 Family Inhibitor
Topics in Medicinal Chemistry
2012
9
28
GlyT-1 Inhibitors: From Hits to Clinical Candidates
Topics in Medicinal Chemistry
2014
9
29
Atypical Elements in Drug Design
Topics in Medicinal Chemistry
2016
9
30
Hsp90 Co-chaperones as Drug Targets in Cancer: Current Perspectives
Topics in Medicinal Chemistry
2016
9
31
Chemical Activation of Sensory TRP Channels
Topics in Medicinal Chemistry
2016
9
32
The Discovery and Development of HCV NS3 Protease Inhibitor Paritaprevir
Topics in Medicinal Chemistry
2019
9
33
Recent Advances in Ion Channel Screening Technologies
Topics in Medicinal Chemistry
2008
8
34
Glycine Transporters and Their Inhibitors
Topics in Medicinal Chemistry
2009
8
35
Improving Solubility via Structural Modification
Topics in Medicinal Chemistry
2013
8
36
Targeting Cellular Cofactors in HIV Therapy
Topics in Medicinal Chemistry
2014
8
37
Computational Docking as a Tool for the Rational Design of Carbohydrate-Based Drugs
Topics in Medicinal Chemistry
2014
8
38
Carbohydrate-Based Anti-Virulence Compounds Against Chronic Pseudomonas aeruginosa Infections with a Focus on Small Molecules
Topics in Medicinal Chemistry
2014
8
39
The Art of Gene Redesign and Recombinant Protein Production: Approaches and Perspectives
Topics in Medicinal Chemistry
2016
8
40
Anti-HIV Agents: Current Status and Recent Trends
Topics in Medicinal Chemistry
2016
8
41
Antibacterial New Target Discovery: Sentinel Examples, Strategies, and Surveying Success
Topics in Medicinal Chemistry
2017
8
42
Messenger RNA as a Novel Therapeutic Approach
Topics in Medicinal Chemistry
2017
8
43
Structure-Based Discovery of Small Molecules Binding to RNA
Topics in Medicinal Chemistry
2017
8
44
Organic Fluorescent Probes for Diagnostics and Bio-Imaging
Topics in Medicinal Chemistry
2019
8
45
The Blood Brain Barrier (BBB)
Topics in Medicinal Chemistry
2014
8
46
Ligand- and Structure-Based Virtual Screening in Drug Discovery
Topics in Medicinal Chemistry
2021
8
47
Taste Receptor Gene Expression Outside the Gustatory System
Topics in Medicinal Chemistry
2014
7
48
The Future of Boron in Medicinal Chemistry: Therapeutic and Diagnostic Applications
Topics in Medicinal Chemistry
2014
7
49
Production of Protein Therapeutics in the Quality by Design (QbD) Paradigm
Topics in Medicinal Chemistry
2016
7
50
The Cyclic Lipopeptide Antibiotics
Topics in Medicinal Chemistry
2017
7
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