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Drug Discovery Today: Technologies
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top-articles
Drug Discovery Today: Technologies
4.0
(top 10%)
impact factor
606
(top 50%)
papers
19.7K
(top 10%)
citations
63
(top 10%)
h
-index
4.2
(top 10%)
impact factor
671
all documents
21.0K
doc citations
116
(top 10%)
g
-index
Top Articles
#
Title
Journal
Year
Citations
1
Lead- and drug-like compounds: the rule-of-five revolution
Drug Discovery Today: Technologies
2004
3,723
2
PROteolysis TArgeting Chimeras (PROTACs) — Past, present and future
Drug Discovery Today: Technologies
2019
458
3
The use of amorphous solid dispersions: A formulation strategy to overcome poor solubility and dissolution rate
Drug Discovery Today: Technologies
2012
436
4
Scaffold hopping
Drug Discovery Today: Technologies
2004
296
5
The production of 3D tumor spheroids for cancer drug discovery
Drug Discovery Today: Technologies
2017
283
6
Vesicles as a tool for transdermal and dermal delivery
Drug Discovery Today: Technologies
2005
259
7
Nanoparticle uptake by the oral route: Fulfilling its potential?
Drug Discovery Today: Technologies
2005
212
8
Clinical trials for BET inhibitors run ahead of the science
Drug Discovery Today: Technologies
2016
209
9
‘In silico’ simulations to assess the ‘in vivo’ consequences of ‘in vitro’ metabolic drug–drug interactions
Drug Discovery Today: Technologies
2004
197
10
Subcutaneous drug delivery and the role of the lymphatics
Drug Discovery Today: Technologies
2005
195
11
A compact review of molecular property prediction with graph neural networks
Drug Discovery Today: Technologies
2020
182
12
Combination of ligand- and structure-based methods in virtual screening
Drug Discovery Today: Technologies
2013
170
13
Ligand efficiency as a guide in fragment hit selection and optimization
Drug Discovery Today: Technologies
2010
167
14
General principles of antibiotic resistance in bacteria
Drug Discovery Today: Technologies
2014
157
15
In silico target fishing: Predicting biological targets from chemical structure
Drug Discovery Today: Technologies
2006
155
16
Prediction of blood–brain barrier permeation in drug discovery from in vivo, in vitro and in silico models
Drug Discovery Today: Technologies
2004
151
17
Multicomponent reactions – opportunities for the pharmaceutical industry
Drug Discovery Today: Technologies
2013
149
18
Overcoming poor oral bioavailability using nanoparticle formulations – opportunities and limitations
Drug Discovery Today: Technologies
2012
144
19
Intracellular delivery of protein and peptide therapeutics
Drug Discovery Today: Technologies
2008
143
20
Multi-objective optimization methods in drug design
Drug Discovery Today: Technologies
2013
134
21
Biofilms as a mechanism of bacterial resistance
Drug Discovery Today: Technologies
2014
130
22
New trends in carbohydrate-based vaccines
Drug Discovery Today: Technologies
2004
123
23
Buccal drug delivery: A challenge already won?
Drug Discovery Today: Technologies
2005
121
24
The controversial world of sirtuins
Drug Discovery Today: Technologies
2014
120
25
Ultrasound-mediated drug delivery to the brain: principles, progress and prospects
Drug Discovery Today: Technologies
2016
120
26
Translational pharmacokinetics and pharmacodynamics of monoclonal antibodies
Drug Discovery Today: Technologies
2016
117
27
Advances in virtual screening
Drug Discovery Today: Technologies
2006
113
28
SNIPERs—Hijacking IAP activity to induce protein degradation
Drug Discovery Today: Technologies
2019
112
29
Advances in screening for membrane permeability: high-resolution PAMPA for medicinal chemists
Drug Discovery Today: Technologies
2004
106
30
Lipid-based formulations for oral delivery of lipophilic drugs
Drug Discovery Today: Technologies
2012
106
31
Chitosan and the mucosal delivery of biotechnology drugs
Drug Discovery Today: Technologies
2005
105
32
Mucoadhesive systems in oral drug delivery
Drug Discovery Today: Technologies
2005
103
33
Smart polymeric micelles for gene and drug delivery
Drug Discovery Today: Technologies
2005
102
34
Nanobodies – from llamas to therapeutic proteins
Drug Discovery Today: Technologies
2010
102
35
Strategies for 3D pharmacophore-based virtual screening
Drug Discovery Today: Technologies
2010
97
36
Conformations and 3D pharmacophore searching
Drug Discovery Today: Technologies
2010
95
37
Alzheimer's disease drug discovery: in vivo screening using Caenorhabditis elegans as a model for β-amyloid peptide-induced toxicity
Drug Discovery Today: Technologies
2013
95
38
Small-molecule PROTAC degraders of the Bromodomain and Extra Terminal (BET) proteins — A review
Drug Discovery Today: Technologies
2019
92
39
Scoring functions for protein–ligand interactions: a critical perspective
Drug Discovery Today: Technologies
2004
91
40
Recent advances in CHO cell line development for recombinant protein production
Drug Discovery Today: Technologies
2020
89
41
Recombinant therapeutic protein production in cultivated mammalian cells: current status and future prospects
Drug Discovery Today: Technologies
2008
88
42
Lipophilicity – beyond octanol/water: a short comparison of modern technologies
Drug Discovery Today: Technologies
2004
86
43
New technologies in computer-aided drug design: Toward target identification and new chemical entity discovery
Drug Discovery Today: Technologies
2006
85
44
Physicochemical profiling: overview of the screens
Drug Discovery Today: Technologies
2004
83
45
Drying methods for protein pharmaceuticals
Drug Discovery Today: Technologies
2008
83
46
Label-free receptor assays
Drug Discovery Today: Technologies
2010
82
47
Overcoming antifungal resistance
Drug Discovery Today: Technologies
2014
80
48
Cereblon modulators: Low molecular weight inducers of protein degradation
Drug Discovery Today: Technologies
2019
77
49
Pharmacophore definition and 3D searches
Drug Discovery Today: Technologies
2004
75
50
Animal models of Alzheimer's disease and drug development
Drug Discovery Today: Technologies
2013
75
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