395
Citations
106
Journals
2012
First Cited
2022
Last Cited

Articles citing This Document (Page 3 of 8)

ArticleJournalYear
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Renal Organic Cation and Anion Transport: From Physiology to Genes☆2014
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In Vitro Kinetic Characterization of Transporter-Mediated PermeabilityAAPS Advances in the Pharmaceutical Sciences Series2013
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Pharmacogenetics of membrane transporters: a review of current approachesMethods in Molecular Biology2014
Prediction of Hepatic Transporter-Mediated Drug–Drug Interaction from In Vitro DataAAPS Advances in the Pharmaceutical Sciences Series2013
The Role of Transporters in Drug Development: Regulatory Science Perspectives from the FDAAAPS Advances in the Pharmaceutical Sciences Series2013
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Evaluation of iberdomide and cytochrome p450 drug-drug interaction potential in vitro and in a phase 1 study in healthy subjectsEuropean Journal of Clinical Pharmacology2021
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Influence of Multidrug Resistance-Associated Proteins on the Excretion of the ABCC1 Imaging Probe 6-Bromo-7-[C]Methylpurine in MiceMolecular Imaging and Biology2019
Lack of Effect of 12-Week Treatment with Risankizumab on the Pharmacokinetics of Cytochrome P450 Probe Substrates in Patients with Moderate to Severe Chronic Plaque PsoriasisClinical Pharmacokinetics2019
Mass Balance and Drug Interaction Potential of Intravenous Eravacycline Administered to Healthy SubjectsAntimicrobial Agents and Chemotherapy2019
Physiologically-Based Pharmacokinetic Models for CYP1A2 Drug-Drug Interaction Prediction: A Modeling Network of Fluvoxamine, Theophylline, Caffeine, Rifampicin, and MidazolamCPT: Pharmacometrics and Systems Pharmacology2019
Effect of CYP3A Inhibition and Induction on the Pharmacokinetics of Suvorexant: Two Phase I, Open-Label, Fixed-Sequence Trials in Healthy SubjectsClinical Drug Investigation2019
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Considerations for Biologic Product Drug-Drug Interactions: A Regulatory PerspectiveClinical Pharmacology and Therapeutics2019
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CYP3A4-mediated effects of rifampicin on the pharmacokinetics of vilaprisan and its UGT1A1-mediated effects on bilirubin glucuronidation in humansBritish Journal of Clinical Pharmacology2018
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A Novel PBPK Modeling Approach to Assess Cytochrome P450 Mediated Drug-Drug Interaction Potential of the Cytotoxic Prodrug EvofosfamideCPT: Pharmacometrics and Systems Pharmacology2018
Drug Interactions With New Synthetic OpioidsFrontiers in Pharmacology2018
Experimental Studies of the Effects of Progesterone on the Functional Activity of P-GlycoproteinPharmaceutical Chemistry Journal2018
Renal Organic Cation and Anion Transport: From Physiology to Genes2018
In Vitro and In Vivo Investigation of Potential for Complex CYP3A Interaction for PF-00251802 (Dagrocorat), a Novel Dissociated Agonist of the Glucocorticoid ReceptorClinical Pharmacology in Drug Development2018
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Drug interactions between non-rifamycin antibiotics and hormonal contraception: a systematic reviewAmerican Journal of Obstetrics and Gynecology2018
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Relationships of Changes in Pharmacokinetic Parameters of Substrate Drugs in Drug-Drug Interactions on Metabolizing Enzymes and TransportersJournal of Clinical Pharmacology2018
Effects of a Fixed-Dose Co-Formulation of Daclatasvir, Asunaprevir, and Beclabuvir on the Pharmacokinetics of a Cocktail of Cytochrome P450 and Drug Transporter Substrates in Healthy SubjectsDrugs in R and D2018
Reverse Translation of US Food and Drug Administration Reviews of Oncology New Molecular Entities Approved in 2011-2017: Lessons Learned for Anticancer Drug DevelopmentClinical and Translational Science2018
In vitro studies and in silico predictions of fluconazole and CYP2C9 genetic polymorphism impact on siponimod metabolism and pharmacokineticsEuropean Journal of Clinical Pharmacology2018
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Effects of Ketoconazole and Rifampicin on the Pharmacokinetics of Nintedanib in Healthy SubjectsEuropean Journal of Drug Metabolism and Pharmacokinetics2018
Disease-Drug Interactions in Inflammatory States via Effects on CYP-Mediated Drug ClearanceJournal of Clinical Pharmacology2018
The Role of Transporters in Drug Accumulation and Mitochondrial Toxicity2018
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Validation of a total IC method which enables in vitro assessment of transporter inhibition under semi-physiological conditionsXenobiotica2017
Selexipag in Pulmonary Arterial Hypertension: Most Updated Evidence From Recent Preclinical and Clinical StudiesJournal of Clinical Pharmacology2017
Unbound liver concentration is the true inhibitor concentration that determines cytochrome P450-mediated drug-drug interactions in rat liverXenobiotica2017
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In vitro metabolism studies of natural products are crucial in the early development of medicinesPhytochemistry Reviews2017
Clarithromycin, Midazolam, and Digoxin: Application of PBPK Modeling to Gain New Insights into Drug-Drug Interactions and Co-medication RegimensAAPS Journal2017
The potential of Epimedium koreanum Nakai for herb-drug interactionJournal of Pharmacy and Pharmacology2017
Systemic clearance and brain distribution of carbazole-based cyanine compounds as Alzheimer's disease drug candidatesScientific Reports2017
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Drug-drug interactions between triazole antifungal agents used to treat invasive aspergillosis and immunosuppressants metabolized by cytochrome P450 3A4Transplant Infectious Disease2017
Boceprevir and Antiretroviral Pharmacokinetic Interactions in HIV/HCV Co-infected Persons: AIDS Clinical Trials Group Study A5309sDrugs in R and D2017
Clinical Pharmacology Considerations for the Development of Immune Checkpoint InhibitorsJournal of Clinical Pharmacology2017
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Assessment of the Drug Interaction Potential of Unconjugated and GalNAc-Conjugated 2'-MOE-ASOsMolecular Therapy - Nucleic Acids2017
Mechanistic in vitro studies confirm that inhibition of the renal apical efflux transporter multidrug and toxin extrusion (MATE) 1, and not altered absorption, underlies the increased metformin exposure observed in clinical interactions with cimetidine, trimethoprim or pyrimethaminePharmacology Research and Perspectives2017
Validation of a microdose probe drug cocktail for clinical drug interaction assessments for drug transporters and CYP3AClinical Pharmacology and Therapeutics2017
Potent inhibition of human organic cation transporter 2 (hOCT2) by β-carboline alkaloidsXenobiotica2017
Inhibition of Intestinal OATP2B1 by the Calcium Receptor Antagonist Ronacaleret Results in a Significant Drug-Drug Interaction by Causing a 2-Fold Decrease in Exposure of RosuvastatinDrug Metabolism and Disposition2017
Effects of Tenapanor on Cytochrome P450-Mediated Drug-Drug InteractionsClinical Pharmacology in Drug Development2017
Angiotensin II Receptor Blockers Inhibit the Generation of Epoxyeicosatrienoic Acid from Arachidonic Acid in Recombinant CYP2C9, CYP2J2 and Human Liver MicrosomesBasic and Clinical Pharmacology and Toxicology2017
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Integrated safety analysis of rolapitant with coadministered drugs from phase II/III trials: an assessment of CYP2D6 or BCRP inhibition by rolapitantAnnals of Oncology2017
Investigating the Additive Interaction of QT-Prolonging Drugs in Older People Using Claims DataDrug Safety2017
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Absorption, Distribution, Metabolism, and Excretion of the Oral Prostaglandin D2 Receptor 2 Antagonist Fevipiprant (QAW039) in Healthy Volunteers and In VitroDrug Metabolism and Disposition2017
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Risk Assessment Using Cytochrome P450 Time-Dependent Inhibition Assays at Single Time and Concentration in the Early Stage of Drug DiscoveryJournal of Pharmaceutical Sciences2017
About P-glycoprotein: a new drugable domain is emerging from structural dataWiley Interdisciplinary Reviews: Computational Molecular Science2017
Tenapanor administration and the activity of the H -coupled transporter PepT1 in healthy volunteersBritish Journal of Clinical Pharmacology2017
Physiologically Based Pharmacokinetic Modeling of Drug Transporters to Facilitate Individualized Dose PredictionJournal of Pharmaceutical Sciences2017
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Drug Interaction Potential of Osilodrostat (LCI699) Based on Its Effect on the Pharmacokinetics of Probe Drugs of Cytochrome P450 Enzymes in Healthy AdultsClinical Drug Investigation2017
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Pharmacokinetic Interactions Between Mirabegron and Metformin, Warfarin, Digoxin or Combined Oral ContraceptivesEuropean Journal of Drug Metabolism and Pharmacokinetics2017
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The Nonmetabolized β-Blocker Nadolol Is a Substrate of OCT1, OCT2, MATE1, MATE2-K, and P-Glycoprotein, but Not of OATP1B1 and OATP1B3Molecular Pharmaceutics2016
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Generation and Characterization of a Breast Cancer Resistance Protein Humanized Mouse ModelMolecular Pharmacology2016