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132 papers • 5,757 citations • Sorted by year • Download PDF (PDF by citations)
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1HECTD3 inhibits NLRP3 inflammasome assembly and activation by blocking NLRP3-NEK7 interaction8.53Citations (PDF)
2<scp>USP3</scp>: Key deubiquitylation enzyme in human diseases
Cancer Science, 2024, 115, 2094-2106
4.00Citations (PDF)
3IL1R2 Blockade Alleviates Immunosuppression and Potentiates Anti-PD-1 Efficacy in Triple-Negative Breast Cancer
Cancer Research, 2024, 84, 2282-2296
0.66Citations (PDF)
4CDK9 targeting PROTAC L055 inhibits ERα-positive breast cancer6.73Citations (PDF)
5Tumor suppressor FRMD3 controls mammary epithelial cell fate determination via notch signaling pathway
Science Advances, 2024, 10,
11.32Citations (PDF)
6PI3K PROTAC overcomes the lapatinib resistance in PIK3CA-mutant HER2 positive breast cancer
Cancer Letters, 2024, 598, 217112
8.52Citations (PDF)
7BRD4-specific PROTAC inhibits basal-like breast cancer partially through downregulating KLF5 expression
Oncogene, 2024, 43, 2914-2926
6.60Citations (PDF)
8Targeting the HECTD3-p62 axis increases the radiosensitivity of triple negative breast cancer cells6.10Citations (PDF)
9TNFAIP2 promotes HIF1α transcription and breast cancer angiogenesis by activating the Rac1-ERK-AP1 signaling axis8.50Citations (PDF)
10Targeting PRMT5 through PROTAC for the treatment of triple-negative breast cancer11.51Citations (PDF)
11RNF126‐Mediated MRE11 Ubiquitination Activates the DNA Damage Response and Confers Resistance of Triple‐Negative Breast Cancer to Radiotherapy
Advanced Science, 2023, 10,
12.822Citations (PDF)
12A novel methuosis inducer DZ-514 possesses antitumor activity via activation of ROS-MKK4-p38 axis in triple negative breast cancer
Cancer Letters, 2023, 555, 216049
8.511Citations (PDF)
13Targeting the KLF5-EphA2 axis can restrain cancer stemness and overcome chemoresistance in basal-like breast cancer8.615Citations (PDF)
14Integrin β4 promotes DNA damage-related drug resistance in triple-negative breast cancer via TNFAIP2/IQGAP1/RAC1
ELife, 2023, 12,
1.63Citations (PDF)
15LncRNA H19 Regulates Breast Cancer DNA Damage Response and Sensitivity to PARP Inhibitors via Binding to ILF24.512Citations (PDF)
16Author Response: Integrin β4 promotes DNA damage-related drug resistance in triple-negative breast cancer via TNFAIP2/IQGAP1/RAC1
2023, ,
0Citations (PDF)
17SGCE promotes breast cancer stemness by promoting the transcription of FGF-BP1 by Sp12.32Citations (PDF)
18Kindlin-2 in myoepithelium controls luminal progenitor commitment to alveoli in mouse mammary gland8.53Citations (PDF)
19YB-1 is a positive regulator of KLF5 transcription factor in basal-like breast cancer
Cell Death and Differentiation, 2022, 29, 1283-1295
13.740Citations (PDF)
20Histone Deacetylase Inhibitors (HDACi) Promote KLF5 Ubiquitination and Degradation in Basal-like Breast Cancer8.615Citations (PDF)
21PRMT5 regulates RNA m6A demethylation for doxorubicin sensitivity in breast cancer
Molecular Therapy, 2022, 30, 2603-2617
10.574Citations (PDF)
22STAMBPL1 promotes breast cancer cell resistance to cisplatin partially by stabilizing MKP-1 expression
Oncogene, 2022, 41, 2265-2274
6.610Citations (PDF)
23Rab13 Sustains Breast Cancer Stem Cells by Supporting Tumor–Stroma Cross-talk
Cancer Research, 2022, 82, 2124-2140
0.615Citations (PDF)
24YB-1 as an Oncoprotein: Functions, Regulation, Post-Translational Modifications, and Targeted Therapy
Cells, 2022, 11, 1217
4.828Citations (PDF)
25A feedforward circuit between KLF5 and lncRNA KPRT4 contributes to basal-like breast cancer
Cancer Letters, 2022, 534, 215618
8.56Citations (PDF)
26Targeting HECTD3-IKKα axis inhibits inflammation-related metastasis26.319Citations (PDF)
27Advances in Biomarkers and Endogenous Regulation of Breast Cancer Stem Cells
Cells, 2022, 11, 2941
4.83Citations (PDF)
28METTL3 acetylation impedes cancer metastasis via fine-tuning its nuclear and cytosolic functions14.143Citations (PDF)
29Progress of Breast Cancer basic research in China8.660Citations (PDF)
30Isochromanoindolenines suppress triple-negative breast cancer cell proliferation partially via inhibiting Akt activation8.63Citations (PDF)
31Glucose-6-phosphate dehydrogenase neutralizes stresses by supporting reductive glutamine metabolism and AMPK activation26.310Citations (PDF)
32Activation of PI3K/AKT/mTOR Pathway Causes Drug Resistance in Breast Cancer4.0218Citations (PDF)
33EphA2: A promising therapeutic target in breast cancer4.436Citations (PDF)
34Targeting ubiquitin conjugating enzyme UbcH5b by a triterpenoid PC3-15 from Schisandra plants sensitizes triple-negative breast cancer cells to lapatinib
Cancer Letters, 2021, 504, 125-136
8.518Citations (PDF)
35Naturally-occurring spinosyn A and its derivatives function as argininosuccinate synthase activator and tumor inhibitor14.137Citations (PDF)
36The roles and regulation of the KLF5 transcription factor in cancers
Cancer Science, 2021, 112, 2097-2117
4.081Citations (PDF)
37Cyst(e)ine in nutrition formulation promotes colon cancer growth and chemoresistance by activating mTORC1 and scavenging ROS26.333Citations (PDF)
38Arginine methyltransferase PRMT5 methylates and stabilizes KLF5 via decreasing its phosphorylation and ubiquitination to promote basal-like breast cancer
Cell Death and Differentiation, 2021, 28, 2931-2945
13.734Citations (PDF)
39Characterization of tree shrew telomeres and telomerase4.42Citations (PDF)
40The methylenetetrahydrofolate reductase (MTHFR) C677T gene polymorphism is associated with breast cancer subtype susceptibility in southwestern China
PLoS ONE, 2021, 16, e0254267
2.54Citations (PDF)
41KAT6A Acetylation of SMAD3 Regulates Myeloid‐Derived Suppressor Cell Recruitment, Metastasis, and Immunotherapy in Triple‐Negative Breast Cancer
Advanced Science, 2021, 8,
12.845Citations (PDF)
42Loss‐of‐Function Genetic Screening Identifies Aldolase A as an Essential Driver for Liver Cancer Cell Growth Under Hypoxia
Hepatology, 2021, 74, 1461-1479
11.674Citations (PDF)
43KLF5-induced lncRNA IGFL2-AS1 promotes basal-like breast cancer cell growth and survival by upregulating the expression of IGFL1
Cancer Letters, 2021, 515, 49-62
8.521Citations (PDF)
44Cancer progression is mediated by proline catabolism in non-small cell lung cancer
Oncogene, 2020, 39, 2358-2376
6.653Citations (PDF)
45Mechanisms of CDK4/6 Inhibitor Resistance in Luminal Breast Cancer4.049Citations (PDF)
46Inhibiting both proline biosynthesis and lipogenesis synergistically suppresses tumor growth8.137Citations (PDF)
47A functional missense variant in ITIH3 affects protein expression and neurodevelopment and confers schizophrenia risk in the Han Chinese population4.411Citations (PDF)
48SGCE Promotes Breast Cancer Stem Cells by Stabilizing EGFR
Advanced Science, 2020, 7,
12.847Citations (PDF)
49Roles of RNF126 and BCA2 E3 ubiquitin ligases in DNA damage repair signaling and targeted cancer therapy
Pharmacological Research, 2020, 155, 104748
9.016Citations (PDF)
50TNF-α increases breast cancer stem-like cells through up-regulating TAZ expression via the non-canonical NF-κB pathway
Scientific Reports, 2020, 10,
3.765Citations (PDF)
51Mifepristone Derivative FZU-00,003 Suppresses Triple-negative Breast Cancer Cell Growth partially via miR-153-KLF5 axis8.614Citations (PDF)
52A new Schiff base copper(II) complex induces cancer cell growth inhibition and apoptosis by multiple mechanisms3.022Citations (PDF)
53Pyrrolo [3,4-b]-quinolin-9-amine compound FZU-0038-056 suppresses triple-negative breast cancer partially through inhibiting the expression of Bcl-2
Aging, 2020, 12, 9621-9632
2.53Citations (PDF)
54Heterogeneity and Subtyping of Triple-Negative Breast Cancer
2020, , 21-40
0Citations (PDF)
55Comprehensive analysis of long noncoding RNAs and mRNAs expression profiles and functional networks during chondrogenic differentiation of murine ATDC5 cells2.02Citations (PDF)
56Glucocorticoid Receptor Signaling Activates TEAD4 to Promote Breast Cancer Progression
Cancer Research, 2019, 79, 4399-4411
0.678Citations (PDF)
57Ilamycin E, a natural product of marine actinomycete, inhibits triple-negative breast cancer partially through ER stress-CHOP-Bcl-28.643Citations (PDF)
58Inhibition of super enhancer downregulates the expression of KLF5 in basal-like breast cancers8.635Citations (PDF)
59USP3 promotes breast cancer cell proliferation by deubiquitinating KLF5
Journal of Biological Chemistry, 2019, 294, 17837-17847
2.353Citations (PDF)
60A thiazole-derived oridonin analogue exhibits antitumor activity by directly and allosterically inhibiting STAT3
Journal of Biological Chemistry, 2019, 294, 17471-17486
2.322Citations (PDF)
61Tumor Suppression of Ras GTPase-Activating Protein RASA5 through Antagonizing Ras Signaling Perturbation in Carcinomas
IScience, 2019, 21, 1-18
3.811Citations (PDF)
62HDAC inhibitors induce proline dehydrogenase (POX) transcription and anti-apoptotic autophagy in triple negative breast cancer2.021Citations (PDF)
63Genetic basis of ruminant headgear and rapid antler regeneration
Science, 2019, 364,
38.2126Citations (PDF)
64The antipsychotic agent flupentixol is a new PI3K inhibitor and potential anticancer drug for lung cancer8.617Citations (PDF)
65CUL7 promotes cancer cell survival through promoting Caspase‐8 ubiquitination
International Journal of Cancer, 2019, 145, 1371-1381
4.519Citations (PDF)
66The role of E3 ubiquitin ligase HECTD3 in cancer and beyond5.622Citations (PDF)
67A novel synthetic ursolic acid derivative inhibits growth and induces apoptosis in breast cancer cell lines1.811Citations (PDF)
68Discovery of novel mifepristone derivatives via suppressing KLF5 expression for the treatment of triple-negative breast cancer5.516Citations (PDF)
69Hypoxia induces miR-153 through the IRE1α-XBP1 pathway to fine tune the HIF1α/VEGFA axis in breast cancer angiogenesis
Oncogene, 2018, 37, 1961-1975
6.6109Citations (PDF)
70Mithramycin A suppresses basal triple-negative breast cancer cell survival partially via down-regulating Krüppel-like factor 5 transcription by Sp13.730Citations (PDF)
71RNF126 as a Biomarker of a Poor Prognosis in Invasive Breast Cancer and CHEK1 Inhibitor Efficacy in Breast Cancer Cells
Clinical Cancer Research, 2018, 24, 1629-1643
6.431Citations (PDF)
72Synthesis and structure–activity relationship studies of MI-2 analogues as MALT1 inhibitors2.714Citations (PDF)
73EZH2 induces the expression of miR-1301 as a negative feedback control mechanism in triple negative breast cancer2.09Citations (PDF)
74miR-153 inhibits the migration and the tube formation of endothelial cells by blocking the paracrine of angiopoietin 1 in breast cancer cells
Angiogenesis, 2018, 21, 849-860
7.444Citations (PDF)
75CC chemokine receptor 7 promotes triple-negative breast cancer growth and metastasis2.015Citations (PDF)
76Krüpple‐like factor 5 is essential for mammary gland development and tumorigenesis
Journal of Pathology, 2018, 246, 497-507
5.225Citations (PDF)
77The roles of <scp>TNFAIP</scp>2 in cancers and infectious diseases4.163Citations (PDF)
78HECTD3 mediates TRAF3 polyubiquitination and type I interferon induction during bacterial infection
Journal of Clinical Investigation, 2018, 128, 4148-4162
9.145Citations (PDF)
79Metformin suppresses triple-negative breast cancer stem cells by targeting KLF5 for degradation
Cell Discovery, 2017, 3,
8.0111Citations (PDF)
80Ursolic acid derivative FZU-03,010 inhibits STAT3 and induces cell cycle arrest and apoptosis in renal and breast cancer cells2.030Citations (PDF)
81Econazole nitrate inhibits PI3K activity and promotes apoptosis in lung cancer cells3.718Citations (PDF)
82YD277 Suppresses Triple-Negative Breast Cancer Partially Through Activating the Endoplasmic Reticulum Stress Pathway
Theranostics, 2017, 7, 2339-2349
11.423Citations (PDF)
83树鼩&amp;mdash;&amp;mdash;作为一种新颖的非人灵长类实验疾病动物模型
Zoological Research, 2017, 38, 127-137
2.754Citations (PDF)
84miR-217 inhibits triple-negative breast cancer cell growth, migration, and invasion through targeting KLF5
PLoS ONE, 2017, 12, e0176395
2.535Citations (PDF)
85Characterization and phylogenetic analysis of Krüppel-like transcription factor (KLF) gene family in tree shrews (<i>Tupaia belangeri chinensis</i>)
Oncotarget, 2017, 8, 16325-16339
1.718Citations (PDF)
86Dexamethasone induces docetaxel and cisplatin resistance partially through up-regulating Krüppel-like factor 5 in triple-negative breast cancer
Oncotarget, 2017, 8, 11555-11565
1.741Citations (PDF)
87Mifepristone Suppresses Basal Triple-Negative Breast Cancer Stem Cells by Down-regulating KLF5 Expression
Theranostics, 2016, 6, 533-544
11.4111Citations (PDF)
88The role of semaphorin 4D in tumor development and angiogenesis in human breast cancer
OncoTargets and Therapy, 2016, Volume 9, 5737-5750
1.628Citations (PDF)
89KHF16 is a Leading Structure from <i>Cimicifuga foetida</i> that Suppresses Breast Cancer Partially by Inhibiting the NF-κB Signaling Pathway
Theranostics, 2016, 6, 875-886
11.432Citations (PDF)
90A new oridonin analog suppresses triple-negative breast cancer cells and tumor growth via the induction of death receptor 5
Cancer Letters, 2016, 380, 393-402
8.552Citations (PDF)
91Generation and characterization of a breast carcinoma model by <scp>PyMT</scp> overexpression in mammary epithelial cells of tree shrew, an animal close to primates in evolution4.533Citations (PDF)
92Transforming growth factor-beta increases breast cancer stem cell population partially through upregulating PMEPA1 expression2.027Citations (PDF)
93Ataxin-3 like (ATXN3L), a member of the Josephin family of deubiquitinating enzymes, promotes breast cancer proliferation by deubiquitinating Krüppel-like factor 5 (KLF5)
Oncotarget, 2015, 6, 21369-21378
1.739Citations (PDF)
94Tobacco carcinogen NNK-induced lung cancer animal models and associated carcinogenic mechanisms2.041Citations (PDF)
95BAP1 promotes breast cancer cell proliferation and metastasis by deubiquitinating KLF514.1152Citations (PDF)
96Hippo pathway in mammary gland development and breast cancer2.053Citations (PDF)
97The interplay between TEAD4 and KLF5 promotes breast cancer partially through inhibiting the transcription of <i>p27</i>Kip1
Oncotarget, 2015, 6, 17685-17697
1.765Citations (PDF)
98Cucurbitacin E Induces Cell Cycle G2/M Phase Arrest and Apoptosis in Triple Negative Breast Cancer
PLoS ONE, 2014, 9, e103760
2.563Citations (PDF)
99Tongshu Capsule Down-Regulates the Expression of Estrogen Receptor α and Suppresses Human Breast Cancer Cell Proliferation
PLoS ONE, 2014, 9, e104261
2.55Citations (PDF)
100PTEN/PIK3CA genes are frequently mutated in spontaneous and medroxyprogesterone acetate-accelerated 7,12-dimethylbenz(a)anthracene-induced mammary tumours of tree shrews
European Journal of Cancer, 2014, 50, 3230-3242
3.319Citations (PDF)
101The HECTD3 E3 Ubiquitin Ligase Suppresses Cisplatin-Induced Apoptosis via Stabilizing MALT1
Neoplasia, 2013, 15, 39-IN15
7.235Citations (PDF)
102RNF115/BCA2 E3 Ubiquitin Ligase Promotes Breast Cancer Cell Proliferation through Targeting p21Waf1/Cip1 for Ubiquitin-Mediated Degradation
Neoplasia, 2013, 15, 1028-1035
7.229Citations (PDF)
103Role of KLF5 in Hormonal Signaling and Breast Cancer Development
Vitamins and Hormones, 2013, , 213-225
0.013Citations (PDF)
104E3 Ubiquitin Ligase RNF126 Promotes Cancer Cell Proliferation by Targeting the Tumor Suppressor p21 for Ubiquitin-Mediated Degradation
Cancer Research, 2013, 73, 385-394
0.659Citations (PDF)
105Krüppel-like Factor 5 Transcription Factor Promotes Microsomal Prostaglandin E2 Synthase 1 Gene Transcription in Breast Cancer
Journal of Biological Chemistry, 2013, 288, 26731-26740
2.339Citations (PDF)
106TAZ antagonizes the WWP1-mediated KLF5 degradation and promotes breast cell proliferation and tumorigenesis
Carcinogenesis, 2012, 33, 59-67
2.982Citations (PDF)
107The Induction of Yes-Associated Protein Expression After Arterial Injury Is Crucial for Smooth Muscle Phenotypic Modulation and Neointima Formation6.293Citations (PDF)
108YAP Promotes Breast Cell Proliferation and Survival Partially through Stabilizing the KLF5 Transcription Factor
American Journal of Pathology, 2012, 180, 2452-2461
3.6105Citations (PDF)
109The WWP1 ubiquitin E3 ligase increases TRAIL resistance in breast cancer
International Journal of Cancer, 2012, 130, 1504-1510
4.526Citations (PDF)
110PMEPA1 promotes androgen receptor‐negative prostate cell proliferation through suppressing the Smad3/4–c‐Myc–p21$^{{\rm Cip1}}$ signaling pathway
Journal of Pathology, 2011, 223, 683-694
5.249Citations (PDF)
111The Induction of KLF5 Transcription Factor by Progesterone Contributes to Progesterone-Induced Breast Cancer Cell Proliferation and Dedifferentiation
Molecular Endocrinology, 2011, 25, 1137-1144
3.649Citations (PDF)
112WWP1: a versatile ubiquitin E3 ligase in signaling and diseases5.696Citations (PDF)
113Reactive oxygen species control senescence‐associated matrix metalloproteinase‐1 through c‐Jun‐N‐terminal kinase4.268Citations (PDF)
114The Fbw7 Tumor Suppressor Targets KLF5 for Ubiquitin-Mediated Degradation and Suppresses Breast Cell Proliferation
Cancer Research, 2010, 70, 4728-4738
0.6129Citations (PDF)
115Regulation of Krüpple-Like Factor 5 by Targeted Protein Degradation0.06Citations (PDF)
116KLF5 Promotes Breast Cell Survival Partially through Fibroblast Growth Factor-binding Protein 1-pERK-mediated Dual Specificity MKP-1 Protein Phosphorylation and Stabilization
Journal of Biological Chemistry, 2009, 284, 16791-16798
2.371Citations (PDF)
117Overexpression of WWP1 is associated with the estrogen receptor and insulin‐like growth factor receptor 1 in breast carcinoma
International Journal of Cancer, 2009, 124, 2829-2836
4.541Citations (PDF)
118Essential role of KLF5 transcription factor in cell proliferation and differentiation and its implications for human diseases5.6220Citations (PDF)
119Proteasomal degradation of the KLF5 transcription factor through a ubiquitin-independent pathway
FEBS Letters, 2007, 581, 1124-1130
2.831Citations (PDF)
120The amplifiedWWP1 gene is a potential molecular target in breast cancer4.5115Citations (PDF)
121The Nedd4-like family of E3 ubiquitin ligases and cancer7.2185Citations (PDF)
122KLF5 promotes cell proliferation and tumorigenesis through gene regulationin the TSU-Pr1 human bladder cancer cell line
International Journal of Cancer, 2006, 118, 1346-1355
4.5127Citations (PDF)
123Genetic and Expression Aberrations of E3 Ubiquitin Ligases in Human Breast Cancer
Molecular Cancer Research, 2006, 4, 695-707
2.952Citations (PDF)
124KLF5 Interacts with p53 in Regulating Survivin Expression in Acute Lymphoblastic Leukemia
Journal of Biological Chemistry, 2006, 281, 14711-14718
2.397Citations (PDF)
125Ubiquitin–proteasome degradation of KLF5 transcription factor in cancer and untransformed epithelial cells
Oncogene, 2005, 24, 3319-3327
6.6120Citations (PDF)
126Human Kruppel-like Factor 5 Is a Target of the E3 Ubiquitin Ligase WWP1 for Proteolysis in Epithelial Cells
Journal of Biological Chemistry, 2005, 280, 41553-41561
2.3120Citations (PDF)
127Regulation of KLF5 involves the Sp1 transcription factor in human epithelial cells
Gene, 2004, 330, 133-142
2.438Citations (PDF)
128<i>KLF5</i> is frequently deleted and down‐regulated but rarely mutated in prostate cancer
Prostate, 2003, 55, 81-88
2.2118Citations (PDF)
129Deletion, Mutation, and Loss of Expression of KLF6 in Human Prostate Cancer
American Journal of Pathology, 2003, 162, 1349-1354
3.6129Citations (PDF)
130A possible tumor suppressor role of the KLF5 transcription factor in human breast cancer
Oncogene, 2002, 21, 6567-6572
6.6130Citations (PDF)
131Defining a common region of deletion at 13q21 in human cancers
Genes Chromosomes and Cancer, 2001, 31, 333-344
3.531Citations (PDF)
132Integrin β4 promotes DNA damage-related drug resistance in triple-negative breast cancer via TNFAIP2/IQGAP1/RAC1
ELife, 0, 12,
1.66Citations (PDF)